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Cyp p450
Cyp p450
paclitaxel tamoxifenul teniposide vinblastin vindesine gefitinib azolice antifungice clotrimazol ketoconazol itraconazol macrolide claritromicin eritromicin Antidepresive triciclice amitriptilin clomipramine imipramin ISRS citalopram escitalopram fluoxetin i norfluoxetine sertralina buspirona ( anxiolitic ) venlafaxin ( SNRI ) Antipsihotice Aripiprazol Haloperidol Risperidona Ziprasidone
puternic / moderat: [12] [13] Inhibitori de proteaz ritonavir [14] indinavir nelfinavir antibiotice macrolide [14] eritromicin telitromicin claritromicin antifungice azolice [14] fluconazol ketoconazol itraconazol nefazodon ( antidepresiv ) bergamottin (constitutive ale grapefruit suc) quercetin ( supliment nutriional ) aprepitant ( antiemetice ) verapamil ( blocant canalelor de calciu ) cloramfenicol ( antibiotic )
puternice: [9] anticonvulsivante , starea de spirit stabilizatori fenitoina ( anticonvulsivant ) carbamazepin [14] oxcarbazepine barbiturice [14] fenobarbital non-nucleozidici ai revers transcriptazei [18] efavirenz nevirapin Etravirina rifampicin [14] ( bactericid ) modafinil ( stimulent ) hyperforin (constitutiv al St Johns Wort ) cyproterone ( antiandrogen , progesteron )
slab: dexametazon ( anti-inflamator , slab imunosupresor ) cimetidin ( antagonist al receptorilor felbamate ( anticonvulsivant ) H2 ) glucocorticoizi ( glucozei din buprenorfin ( analgezic ) snge crete, imunosupresoare ) cafestol (n cafea nefiltrat) griseofulvina ( antifungic ) pioglitazon ( hipoglicemica ) nespecificat: [13] primidona ( anticonvulsivant ) amiodarona ( antiaritmice ) topiramat ( anticonvulsivant ) ciprofloxacina (antibiotic) troglitazone ( hipoglicemica ) ciclosporin ( imunosupresoare) rifabutin (n tuberculoz ) diltiazem ( blocant canalelor de calciu ) imatinib ( anticanceroase ) Echinacea ( imunostimulator ) enoxacin ( antibacteriene ) ergotamin (n migren ) metronidazol ( antibacteriene ) mifepristonul ( abortive ) norfloxacin (antibiotic) tofisopam ( anxiolitic ) non-nucleozidici ai revers transcriptazei [18] delavirdin efavirenz
Opiacee analgezice alfentanil codeina fentanil metadon Benzodiazepine alprazolam Clonazepam flunitrazepam midazolam triazolam Statine atorvastatin lovastatin simvastatin Blocante ale canalelor de calciu amlodipin diltiazem felodipin nifedipin verapamilul Amiodarona ( antiaritmice ) Inhibitori ai PDE5 sildenafil Kinins ( vasodilatatoare , musculaturii netede contractori) Hormonilor sexuali agonitii i antagonitii estradiol ( estrogen ) etinilestradiol ( contraceptive hormonale ) Finasteride ( antiandrogen) levonorgestrel ( hormon sexual feminin , contraceptive orale ) mifepristonul (antiprogesterone , antiimplantare agent) testosteron ( androgeni ) toremifen ( SERM ) Astemizol ( antagonist H1 , antipruriginoas ) Warfarina ( anticoagulant ) minore:
nevirapin gestodene ( contraceptive hormonale ) mibefradil (n angin pectoral ) inhibitori de proteaz saquinavir ISRS fluoxetina / norfluoxetine fluvoxamina fructe stele [19] piperine lapte de ciulini [20]