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Effect: Initial depolarization causes transient contractions, followed by prolonged flaccid paralysis depolarization is then followed by repolarization that is also accompanied by paralysis
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especially at neuromuscular junctions. Effect: Prevents depolarization by ACh, causes flaccid paralysis can cause histamine release with hypotension weak block of cardiac muscarinic ACh receptors
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especially at neuromuscular junctions. Effect: Prevents depolarization by ACh, causes flaccid paralysis.
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Pharmacokinetics, Interactions : Not dependent on renal or hepatic function duration, ~2545 min Toxicities :
prolonged apnea.(less toxic than previous).
especially at neuromuscular junctions. Effect: Prevents depolarization by ACh, causes flaccid paralysis. slight antimuscarinic effect.
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impairment.
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inhibition of motor neurons. Effect: Pre- and postsynaptic inhibition of motor output.
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stretch reflex in spinal cord. Effect: Reduction in hyperactive muscle reflexes antimuscarinic effects.
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Orphenadrine.
others: Like cyclobenzaprine with varying degrees of antimuscarinic effect
central nervous system. Effect: Increases interneuron inhibition of primary motor afferents in spinal cord central sedation.
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cerebral palsy. Stroke. spinal cord injury. acute spasm due to:
muscle injury
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Pharmacokinetics, Interactions :
oral duration, 46 h . Toxicities :
Muscle weakness .
IV,
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