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MIMS Summary Table

DRUGS TO AVOID IN G6PD DEFICIENCY


DEFINITE RISK OF HAEMOLYSIS POSSIBLE RISK OF HAEMOLYSIS

G6PD Deficiency
Pharmacological Drugs* Pharmacological Drugs*
Class Class
Anthelmintics • ß-Naphthol Analgesics • Acetylsalicylic acid
• Niridazole (Aspirin)
• Stibophen • Acetanilide
• Paracetamol
Antibiotics • Nitrofurans (Acetaminophen)
- Nitrofurantoin • Aminophenazone
- Nitrofurazone (Aminopyrine)
• Quinolones • Dipyrone
- Ciprofloxacin (Metamizole)
- Moxifloxacin • Phenacetin
- Nalidixic acid • Phenazone
- Norfloxacin (Antipyrine)
- Ofloxacin • Phenylbutazone
• Chloramphenicol • Tiaprofenic acid
• Sulfonamides
- Co-trimoxazole Antibiotics • Furazolidone
(Sulfamethoxazole + • Streptomycin
Trimethoprim) • Sulfonamides
- Sulfacetamide - Sulfacytine
- Sulfadiazine - Sulfaguanidine
- Sulfadimidine - Sulfamerazine
- Sulfamethoxazole - Sulfamethoxypyridazole
- Sulfanilamide Anticonvulsants • Phenytoin
- Sulfapyridine
- Sulfasalazine Antidiabetics • Glibenclamide
(Salazosulfapyridine)
- Sulfisoxazole Antidotes • Dimercaprol (BAL)
(Sulfafurazole) Antihistamines • Antazoline (Antistine)
• Diphenhydramine
Antimalarials • Mepacrine • Tripelennamine
• Pamaquine
• Pentaquine Antihypertensives • Hydralazine
• Primaquine • Methyldopa
Antimethemo- • Methylene blue Antimalarials • Chloroquine & derivatives
globinaemic Agents • Proguanil
• Pyrimethamine
Antimycobacterials • Dapsone • Quinidine
• Para-aminosalicylic acid • Quinine
• Sulfones
- Aldesulfone sodium Antimycobacterials • Isoniazid
(Sulfoxone)
- Glucosulfone Antiparkinsonism Agents • Trihexyphenidyl
- Thiazosulfone (Benzhexol)

Antineoplastic Adjuncts • Doxorubicin Cardiovascular Drugs • Dopamine (L-dopa)


• Rasburicase • Procainamide
• Quinidine
Genitourinary Analgesics • Phenazopyridine Diagnostic Agent • Toluidine blue
(Pyridium) for Cancer Detection
Others • Acetylphenylhydrazine Gout Preparations • Colchicine
• Phenylhydrazine • Probenecid
Hormonal Contraceptives • Mestranol
Nitrates • Isobutyl nitrite
Vitamin K Substance • Menadiol Na sulfate
• Menadione
• Menadione Na bisulfite
• Phytomenadione
Vitamins • Ascorbic acid (Vit C)
(rare)
Others • Arsine
• Berberine
(in Coptis chinensis)
• Fava beans
• Naphthalene
(in mothballs)
• Para-aminobenzoic acid
*Nomenclature based on INN (International non-proprietary name)
Refer to www.g6pd.org for further information.
Please refer to the Contents page for more Summary Tables.

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Copyright © 2006 MIMS

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